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Ipamorelin Monotherapy Protocol

Published August 27, 2026 1 min read 2 mg Popular

Overview

Ipamorelin is a pentapeptide GH secretagogue and ghrelin receptor agonist. It is highly selective for GH release u2014 unlike GHRP-2 or GHRP-6, it does not significantly elevate cortisol, aldosterone, or prolactin at standard doses. Best administered pre-bed to coincide with natural GH secretion.

Dosing & Reconstitution Guide

Once daily (pre-bed) u00b7 200u2013300 mcg u00b7 Half-life: ~2 hr

Reconstitution Table (2 mL mL BAC water u2192 2 mg)

Phase Dose Draw (U-100)
Starting dose 100 mcg 1 Unit
Standard dose 200u2013300 mcg 2u20133 Units

Reconstitute 2 mg with 2 mL BAC water u2192 1,000 mcg/mL. Inject SC 30u201360 min before sleep. Avoid carbohydrates 2 hours before injection (blunts GH pulse).

Ipamorelin does not cause cortisol spikes typical of older GHRPs. Still, extended use should be cycled (e.g. 12 weeks on, 4 weeks off). Research use only.

Potential Benefits & Side Effects

Potential Benefits

  • Clean GH pulse without cortisol elevation
  • Improved sleep quality and recovery
  • Lean body mass support
  • Bone density maintenance
  • Anti-aging potential through IGF-1 axis

Possible Side Effects

  • Water retention at higher doses
  • Mild headache (initial use)
  • Mild injection-site redness

Storage Instructions

Lyophilized Powder

  • Short-term (<3 months): Refrigerate at 2u00b0Cu20138u00b0C
  • Long-term: Freeze at u221220u00b0C or lower
  • Protect from light and moisture
  • Allow vial to reach room temperature before opening

Reconstituted Solution

  • Refrigerate at 2u00b0Cu20138u00b0C u2014 do not freeze
  • Use within 28 days when reconstituted with BAC water
  • Always use sterile technique when drawing doses

References

Raun K. et al. (1998)

Ipamorelin u2014 a new GH-releasing peptide with no effect on motilin

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Important Note

This protocol guide is for educational and research purposes only. It is not medical advice. Always consult a qualified healthcare professional before using any peptide compound.